Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with all data for entry = 50036745
TargetBifunctional purine biosynthesis protein ATIC(Homo sapiens (Human))
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50369444(CHEMBL608337)
Affinity DataIC50:  125nMAssay Description:Inhibitory activity against AICAR formyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional purine biosynthesis protein ATIC(Homo sapiens (Human))
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50080319(10-Formyl-8-deazafolic acid | CHEMBL114215)
Affinity DataIC50:  6.40E+3nMAssay Description:Inhibitory activity against AICAR formyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional purine biosynthesis protein ATIC(Homo sapiens (Human))
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM22579(AICAR | Aminoimidazole-4-carboxamide ribonucleotid...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibitory activity against AICAR formyltransferaseMore data for this Ligand-Target Pair
TargetBifunctional purine biosynthesis protein ATIC(Homo sapiens (Human))
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50080320((2R)-2-{[4-(N-{[(6R)-2-amino-4-oxo-1,4,4a,5,6,7,8,...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibitory activity against AICAR formyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional purine biosynthesis protein ATIC(Homo sapiens (Human))
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50369444(CHEMBL608337)
Affinity DataKd:  20nMAssay Description:Binding affinity towards AICAR formyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed