Compile Data Set for Download or QSAR
maximum 50k data
Found 19 Enz. Inhib. hit(s) with all data for entry = 50042900
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50432927(CHEMBL2377219)
Affinity DataEC50:  604nMAssay Description:Inhibition of 11beta-HSD1 in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM29860(N-(Pyridin-2-yl) arylsulfonamide, 22)
Affinity DataEC50:  53nMAssay Description:Inhibition of 11beta-HSD1 in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50432929(CHEMBL2377217)
Affinity DataEC50:  936nMAssay Description:Inhibition of 11beta-HSD1 in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50432930(CHEMBL2377216)
Affinity DataEC50:  51nMAssay Description:Inhibition of 11beta-HSD1 in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50432931(CHEMBL2377215)
Affinity DataEC50:  1.16E+3nMAssay Description:Inhibition of 11beta-HSD1 in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50432932(CHEMBL2377214)
Affinity DataEC50:  184nMAssay Description:Inhibition of 11beta-HSD1 in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50432931(CHEMBL2377215)
Affinity DataEC50:  327nMAssay Description:Inhibition of 11beta-HSD1 in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50432933(CHEMBL2377212)
Affinity DataEC50:  58nMAssay Description:Inhibition of 11beta-HSD1 in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM29866(N-(Pyridin-2-yl) arylsulfonamide, 28)
Affinity DataEC50:  10nMAssay Description:Inhibition of 11beta-HSD1 in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50432934(CHEMBL2377211)
Affinity DataEC50:  49nMAssay Description:Inhibition of 11beta-HSD1 in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50432935(CHEMBL2377210)
Affinity DataEC50:  72nMAssay Description:Inhibition of 11beta-HSD1 in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50432936(CHEMBL2377209)
Affinity DataEC50:  0.0300nMAssay Description:Inhibition of 11beta-HSD1 in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50432937(CHEMBL2377208)
Affinity DataEC50:  194nMAssay Description:Inhibition of 11beta-HSD1 in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50432938(CHEMBL2377207)
Affinity DataEC50:  1.98E+3nMAssay Description:Inhibition of 11beta-HSD1 in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50432939(CHEMBL2377206)
Affinity DataEC50:  213nMAssay Description:Inhibition of 11beta-HSD1 in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50432940(CHEMBL2377205)
Affinity DataEC50:  21nMAssay Description:Inhibition of 11beta-HSD1 in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50432941(CHEMBL2377204)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of 11beta-HSD1 in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM29864(N-(Pyridin-2-yl) arylsulfonamide, 26)
Affinity DataEC50:  5nMAssay Description:Inhibition of 11beta-HSD1 in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50432928(CHEMBL2377218)
Affinity DataEC50:  423nMAssay Description:Inhibition of 11beta-HSD1 in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed