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Found 11 Enz. Inhib. hit(s) with all data for entry = 50017979
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Guang Xi University Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50606662(CHEMBL5221129)
Affinity DataKi:  2.30nMAssay Description:Inhibition of MCT1 in rat erythrocytesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLarge neutral amino acids transporter small subunit 1(Homo sapiens (Human))
Guang Xi University Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50606667(CHEMBL5220432)
Affinity DataKi:  2.10E+6nMAssay Description:Competitive inhibition of human LAT1 expressed in HEK293 cells assessed as inhibition of L-[14C]-Leucine uptake by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMonocarboxylate transporter 4(Homo sapiens (Human))
Guang Xi University Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50606665(Isotense | Londomin | NSC-77030 | Neoreserpan | SU...)
Affinity DataIC50:  1nMAssay Description:Inhibition of MCT4 in human NCI-H358 cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMonocarboxylate transporter 4(Homo sapiens (Human))
Guang Xi University Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50606665(Isotense | Londomin | NSC-77030 | Neoreserpan | SU...)
Affinity DataIC50:  1nMAssay Description:Inhibition of MCT4 in human MDA-MB-231 cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMonocarboxylate transporter 4(Homo sapiens (Human))
Guang Xi University Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50606664(CHEMBL1616099)
Affinity DataIC50:  1nMAssay Description:Inhibition of MCT4 in human MDA-MB-231 cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMonocarboxylate transporter 4(Homo sapiens (Human))
Guang Xi University Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50606663(CHEMBL5219543)
Affinity DataIC50:  1nMAssay Description:Inhibition of MCT4 in human NCI-H358 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMonocarboxylate transporter 4(Homo sapiens (Human))
Guang Xi University Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50606664(CHEMBL1616099)
Affinity DataIC50:  1nMAssay Description:Inhibition of MCT4 in human NCI-H358 cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMonocarboxylate transporter 4(Homo sapiens (Human))
Guang Xi University Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50606663(CHEMBL5219543)
Affinity DataIC50:  1nMAssay Description:Inhibition of MCT4 in human MDA-MB-231 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Guang Xi University Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50606661(CHEMBL5220706)
Affinity DataIC50:  66nMAssay Description:Inhibition of MCT1 in rat RBE4 cells assessed as reduction in [14C]lactate uptake measured after 15 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Guang Xi University Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM4350((2E)-2-cyano-3-(4-hydroxyphenyl)prop-2-enoic acid ...)
Affinity DataIC50:  281nMAssay Description:Inhibition of MCT1 in rat RBE4 cells assessed as reduction in [14C]lactate uptake measured after 15 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetLarge neutral amino acids transporter small subunit 1(Homo sapiens (Human))
Guang Xi University Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50606666(CHEMBL5219332)
Affinity DataIC50:  1.82E+4nMAssay Description:Inhibition of LAT1 in human MCF7 cells assessed as inhibition of leucine uptakeMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed