Compile Data Set for Download or QSAR
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Found 23 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 2171
TargetMonocarboxylate transporter 4(Homo sapiens (Human))
Vettore

US Patent
LigandPNGBDBM345267(2-[[1-[(2-Chlorophenyl)methyl]-5-[3- (trifluorome...)
Affinity DataIC50:  20nMAssay Description:MCT4 may be stably expressed in MDA-MB-453 breast cancer cells that do not express native MCT1 or MCT4. MCT4 activity may be assessed by monitoring t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))
Vettore

US Patent
LigandPNGBDBM345264(2-[[5-(3-Chlorophenyl)-1-[(2- chlorophenyl)methyl...)
Affinity DataIC50:  21nMAssay Description:MCT4 may be stably expressed in MDA-MB-453 breast cancer cells that do not express native MCT1 or MCT4. MCT4 activity may be assessed by monitoring t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))
Vettore

US Patent
LigandPNGBDBM345268(2-[[1-[(2-Chlorophenyl)methyl]-5-(3- methoxypheny...)
Affinity DataIC50:  26nMAssay Description:MCT4 may be stably expressed in MDA-MB-453 breast cancer cells that do not express native MCT1 or MCT4. MCT4 activity may be assessed by monitoring t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))
Vettore

US Patent
LigandPNGBDBM345266(2-[[1-[(2-Chlorophenyl)methyl]-5-(3- fluorophenyl...)
Affinity DataIC50:  38nMAssay Description:MCT4 may be stably expressed in MDA-MB-453 breast cancer cells that do not express native MCT1 or MCT4. MCT4 activity may be assessed by monitoring t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))
Vettore

US Patent
LigandPNGBDBM345265(2-[[1-[(2-Chlorophenyl)methyl]-5-(m- tolyl)pyrazo...)
Affinity DataIC50:  45nMAssay Description:MCT4 may be stably expressed in MDA-MB-453 breast cancer cells that do not express native MCT1 or MCT4. MCT4 activity may be assessed by monitoring t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))
Vettore

US Patent
LigandPNGBDBM345258(2-[[1-[(2-Chlorophenyl)methyl]-5-(4- fluorophenyl...)
Affinity DataIC50:  68nMAssay Description:MCT4 may be stably expressed in MDA-MB-453 breast cancer cells that do not express native MCT1 or MCT4. MCT4 activity may be assessed by monitoring t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))
Vettore

US Patent
LigandPNGBDBM345262(2-[[1-[(2-Chlorophenyl)methyl]-5-phenyl- pyrazol-...)
Affinity DataIC50:  69nMAssay Description:MCT4 may be stably expressed in MDA-MB-453 breast cancer cells that do not express native MCT1 or MCT4. MCT4 activity may be assessed by monitoring t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))
Vettore

US Patent
LigandPNGBDBM345257(2-[[5-(4-Chlorophenyl)-1-[(2- chlorophenyl)methyl...)
Affinity DataIC50:  72nMAssay Description:MCT4 may be stably expressed in MDA-MB-453 breast cancer cells that do not express native MCT1 or MCT4. MCT4 activity may be assessed by monitoring t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))
Vettore

US Patent
LigandPNGBDBM345273(2-[[5-(4-Chlorophenyl)-1-[(2- fluorophenyl)methyl...)
Affinity DataIC50:  110nMAssay Description:MCT4 may be stably expressed in MDA-MB-453 breast cancer cells that do not express native MCT1 or MCT4. MCT4 activity may be assessed by monitoring t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))
Vettore

US Patent
LigandPNGBDBM345272(2-[[1-[(2-Chlorophenyl)methyl]-5-thiazol- 2-yl-py...)
Affinity DataIC50:  152nMAssay Description:MCT4 may be stably expressed in MDA-MB-453 breast cancer cells that do not express native MCT1 or MCT4. MCT4 activity may be assessed by monitoring t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))
Vettore

US Patent
LigandPNGBDBM345259(2-[[5-(4-Chlorophenyl)-1-[(2,4- dichlorophenyl)me...)
Affinity DataIC50:  160nMAssay Description:MCT4 may be stably expressed in MDA-MB-453 breast cancer cells that do not express native MCT1 or MCT4. MCT4 activity may be assessed by monitoring t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))
Vettore

US Patent
LigandPNGBDBM345260(2-[[5-(4-Chlorophenyl)-1-[(2,4- dichlorophenyl)me...)
Affinity DataIC50:  201nMAssay Description:MCT4 may be stably expressed in MDA-MB-453 breast cancer cells that do not express native MCT1 or MCT4. MCT4 activity may be assessed by monitoring t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))
Vettore

US Patent
LigandPNGBDBM345277(2-[[5-(4-Chlorophenyl)-1-(3- pyridylmethyl)pyrazo...)
Affinity DataIC50:  250nMAssay Description:MCT4 may be stably expressed in MDA-MB-453 breast cancer cells that do not express native MCT1 or MCT4. MCT4 activity may be assessed by monitoring t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))
Vettore

US Patent
LigandPNGBDBM345263(2-[[5-(2-Chlorophenyl)-1-[(2- chlorophenyl)methyl...)
Affinity DataIC50:  320nMAssay Description:MCT4 may be stably expressed in MDA-MB-453 breast cancer cells that do not express native MCT1 or MCT4. MCT4 activity may be assessed by monitoring t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))
Vettore

US Patent
LigandPNGBDBM356632(US10214492, Example 1 | US11292767, Example 1)
Affinity DataIC50:  340nMAssay Description:MCT4 may be stably expressed in MDA-MB-453 breast cancer cells that do not express native MCT1 or MCT4. MCT4 activity may be assessed by monitoring t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))
Vettore

US Patent
LigandPNGBDBM345271(1-[[5-(4-Chlorophenyl)-1-[(2- chlorophenyl)methyl...)
Affinity DataIC50:  440nMAssay Description:MCT4 may be stably expressed in MDA-MB-453 breast cancer cells that do not express native MCT1 or MCT4. MCT4 activity may be assessed by monitoring t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))
Vettore

US Patent
LigandPNGBDBM345256(2-[[5-(4-Chlorophenyl)-1-[(4- chlorophenyl)methyl...)
Affinity DataIC50:  450nMAssay Description:MCT4 may be stably expressed in MDA-MB-453 breast cancer cells that do not express native MCT1 or MCT4. MCT4 activity may be assessed by monitoring t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))
Vettore

US Patent
LigandPNGBDBM345261(2-[[1-Benzyl-5-(4-Chlorophenyl)pyrazol- 3-yl]meth...)
Affinity DataIC50:  720nMAssay Description:MCT4 may be stably expressed in MDA-MB-453 breast cancer cells that do not express native MCT1 or MCT4. MCT4 activity may be assessed by monitoring t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))
Vettore

US Patent
LigandPNGBDBM345269(2-[[1-[(2-Chlorophenyl)methyl]-5- cyclohexyl-pyra...)
Affinity DataIC50:  900nMAssay Description:MCT4 may be stably expressed in MDA-MB-453 breast cancer cells that do not express native MCT1 or MCT4. MCT4 activity may be assessed by monitoring t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))
Vettore

US Patent
LigandPNGBDBM345270(2-[[1-[(2-Chlorophenyl)methyl]-5- cyclopentyl-pyr...)
Affinity DataIC50:  1.00E+3nMAssay Description:MCT4 may be stably expressed in MDA-MB-453 breast cancer cells that do not express native MCT1 or MCT4. MCT4 activity may be assessed by monitoring t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))
Vettore

US Patent
LigandPNGBDBM345276(2-[[5-(4-Chlorophenyl)-1-(2- pyridylmethyl)pyrazo...)
Affinity DataIC50:  1.40E+4nMAssay Description:MCT4 may be stably expressed in MDA-MB-453 breast cancer cells that do not express native MCT1 or MCT4. MCT4 activity may be assessed by monitoring t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))
Vettore

US Patent
LigandPNGBDBM345257(2-[[5-(4-Chlorophenyl)-1-[(2- chlorophenyl)methyl...)
Affinity DataIC50:  1.70E+4nMAssay Description:MCT4 may be stably expressed in MDA-MB-453 breast cancer cells that do not express native MCT1 or MCT4. MCT4 activity may be assessed by monitoring t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonocarboxylate transporter 4(Homo sapiens (Human))
Vettore

US Patent
LigandPNGBDBM345275(2-[[5-(4-chlorophenyl)-1-(4- pyridylmethyl)pyrazo...)
Affinity DataIC50:  3.50E+4nMAssay Description:MCT4 may be stably expressed in MDA-MB-453 breast cancer cells that do not express native MCT1 or MCT4. MCT4 activity may be assessed by monitoring t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent