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Found 6 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50031661
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316849(2-(4-Fluorobenzyl)-5,6-dimethyl-3-prop-2-yn-1-ylth...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316851(2-Phenyl-3-prop-2-yn-1-yl-3,5,6,7-tetrahydro-4H-cy...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316850(2-Methyl-3-prop-2-yn-1-yl-3,5,6,7-tetrahydro-4H-cy...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316847(2,5,6-Trimethyl-3-prop-2-yn-1-ylthieno[2,3-d]pyrim...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Institute Of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50316846(2-(4-Fluorobenzyl)-3-prop-2-yn-1-yl-5,6,7,8-tetrah...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed