TargetDihydrofolate reductase(Homo sapiens (Human))
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Affinity DataKi: 4.5nMAssay Description:Inhibition of human DHFR assessed as oxidation of NADPH using dihydrofolate as substrate pre-incubated for 10 mins before substrate addition by spect...More data for this Ligand-Target Pair
TargetDihydrofolate reductase(Homo sapiens (Human))
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Affinity DataKi: 5.80nMAssay Description:Inhibition of human DHFR assessed as oxidation of NADPH using dihydrofolate as substrate pre-incubated for 10 mins before substrate addition by spect...More data for this Ligand-Target Pair
TargetDihydrofolate reductase(Homo sapiens (Human))
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Affinity DataKi: 10.1nMAssay Description:Inhibition of human DHFR assessed as oxidation of NADPH using dihydrofolate as substrate pre-incubated for 10 mins before substrate addition by spect...More data for this Ligand-Target Pair
TargetDihydrofolate reductase(Homo sapiens (Human))
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Affinity DataKi: 11.1nMAssay Description:Inhibition of human DHFR assessed as oxidation of NADPH using dihydrofolate as substrate pre-incubated for 10 mins before substrate addition by spect...More data for this Ligand-Target Pair
TargetDihydrofolate reductase(Homo sapiens (Human))
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Affinity DataKi: 11.1nMAssay Description:Inhibition of human DHFR assessed as oxidation of NADPH using dihydrofolate as substrate pre-incubated for 10 mins before substrate addition by spect...More data for this Ligand-Target Pair
TargetDihydrofolate reductase(Homo sapiens (Human))
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Inhibition of human DHFR assessed as oxidation of NADPH using dihydrofolate as substrate pre-incubated for 10 mins before substrate addition by spect...More data for this Ligand-Target Pair
TargetDihydrofolate reductase(Homo sapiens (Human))
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Affinity DataKi: 12.2nMAssay Description:Inhibition of human DHFR assessed as oxidation of NADPH using dihydrofolate as substrate pre-incubated for 10 mins before substrate addition by spect...More data for this Ligand-Target Pair
TargetDihydrofolate reductase(Homo sapiens (Human))
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Affinity DataKi: 20.9nMAssay Description:Inhibition of human DHFR assessed as oxidation of NADPH using dihydrofolate as substrate pre-incubated for 10 mins before substrate addition by spect...More data for this Ligand-Target Pair
TargetDihydrofolate reductase(Homo sapiens (Human))
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Affinity DataKi: 22.2nMAssay Description:Inhibition of human DHFR assessed as oxidation of NADPH using dihydrofolate as substrate pre-incubated for 10 mins before substrate addition by spect...More data for this Ligand-Target Pair
TargetDihydrofolate reductase(Homo sapiens (Human))
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Affinity DataKi: 26.3nMAssay Description:Inhibition of human DHFR assessed as oxidation of NADPH using dihydrofolate as substrate pre-incubated for 10 mins before substrate addition by spect...More data for this Ligand-Target Pair
TargetDihydrofolate reductase(Homo sapiens (Human))
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Affinity DataKi: 27.5nMAssay Description:Inhibition of human DHFR assessed as oxidation of NADPH using dihydrofolate as substrate pre-incubated for 10 mins before substrate addition by spect...More data for this Ligand-Target Pair
TargetDihydrofolate reductase(Homo sapiens (Human))
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Affinity DataKi: 34nMAssay Description:Inhibition of human DHFR assessed as oxidation of NADPH using dihydrofolate as substrate pre-incubated for 10 mins before substrate addition by spect...More data for this Ligand-Target Pair
TargetDihydrofolate reductase(Homo sapiens (Human))
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Affinity DataKi: 41.1nMAssay Description:Inhibition of human DHFR assessed as oxidation of NADPH using dihydrofolate as substrate pre-incubated for 10 mins before substrate addition by spect...More data for this Ligand-Target Pair
TargetDihydrofolate reductase(Homo sapiens (Human))
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Affinity DataKi: 44.1nMAssay Description:Inhibition of human DHFR assessed as oxidation of NADPH using dihydrofolate as substrate pre-incubated for 10 mins before substrate addition by spect...More data for this Ligand-Target Pair
TargetDihydrofolate reductase(Homo sapiens (Human))
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Affinity DataKi: 85nMAssay Description:Inhibition of human DHFR assessed as oxidation of NADPH using dihydrofolate as substrate pre-incubated for 10 mins before substrate addition by spect...More data for this Ligand-Target Pair
TargetDihydrofolate reductase(Homo sapiens (Human))
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Affinity DataKi: 95.6nMAssay Description:Inhibition of human DHFR assessed as oxidation of NADPH using dihydrofolate as substrate pre-incubated for 10 mins before substrate addition by spect...More data for this Ligand-Target Pair
TargetDihydrofolate reductase(Homo sapiens (Human))
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Affinity DataKi: 129nMAssay Description:Inhibition of human DHFR assessed as oxidation of NADPH using dihydrofolate as substrate pre-incubated for 10 mins before substrate addition by spect...More data for this Ligand-Target Pair
TargetDihydrofolate reductase(Homo sapiens (Human))
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Affinity DataKi: 138nMAssay Description:Inhibition of human DHFR assessed as oxidation of NADPH using dihydrofolate as substrate pre-incubated for 10 mins before substrate addition by spect...More data for this Ligand-Target Pair
TargetDihydrofolate reductase(Homo sapiens (Human))
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Affinity DataKi: 245nMAssay Description:Inhibition of human DHFR assessed as oxidation of NADPH using dihydrofolate as substrate pre-incubated for 10 mins before substrate addition by spect...More data for this Ligand-Target Pair
TargetDihydrofolate reductase(Homo sapiens (Human))
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Affinity DataKi: 253nMAssay Description:Inhibition of human DHFR assessed as oxidation of NADPH using dihydrofolate as substrate pre-incubated for 10 mins before substrate addition by spect...More data for this Ligand-Target Pair
TargetDihydrofolate reductase(Homo sapiens (Human))
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Affinity DataKi: 323nMAssay Description:Inhibition of human DHFR assessed as oxidation of NADPH using dihydrofolate as substrate pre-incubated for 10 mins before substrate addition by spect...More data for this Ligand-Target Pair
TargetDihydrofolate reductase(Homo sapiens (Human))
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Affinity DataKi: 702nMAssay Description:Inhibition of human DHFR assessed as oxidation of NADPH using dihydrofolate as substrate pre-incubated for 10 mins before substrate addition by spect...More data for this Ligand-Target Pair
TargetDihydrofolate reductase(Homo sapiens (Human))
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Affinity DataKi: 743nMAssay Description:Inhibition of human DHFR assessed as oxidation of NADPH using dihydrofolate as substrate pre-incubated for 10 mins before substrate addition by spect...More data for this Ligand-Target Pair
TargetDihydrofolate reductase(Homo sapiens (Human))
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Affinity DataKi: 775nMAssay Description:Inhibition of human DHFR assessed as oxidation of NADPH using dihydrofolate as substrate pre-incubated for 10 mins before substrate addition by spect...More data for this Ligand-Target Pair
TargetDihydrofolate reductase(Homo sapiens (Human))
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Affinity DataKi: 1.14E+3nMAssay Description:Inhibition of human DHFR assessed as oxidation of NADPH using dihydrofolate as substrate pre-incubated for 10 mins before substrate addition by spect...More data for this Ligand-Target Pair
TargetDihydrofolate reductase(Homo sapiens (Human))
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Trius Therapeutics, San Diego, Ca 92121, United States.
Curated by ChEMBL
Affinity DataKi: 1.91E+4nMAssay Description:Inhibition of human DHFR assessed as oxidation of NADPH using dihydrofolate as substrate pre-incubated for 10 mins before substrate addition by spect...More data for this Ligand-Target Pair