Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 50035143
TargetMetabotropic glutamate receptor 3(Rattus norvegicus (Rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50052398((2R,4R)-4-aminopyrrolidine-2,4-dicarboxylic acid |...)
Affinity DataEC50:  1.70E+3nMAssay Description:Effective concentration required for agonistic activity at Metabotropic glutamate receptor 3More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 3(Rattus norvegicus (Rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50102116((2R,4R)-4-amino-1-(2-nitrobenzyl)pyrrolidine-2,4-d...)
Affinity DataEC50:  6.80E+3nMAssay Description:Effective concentration required for agonistic activity at Metabotropic glutamate receptor 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 3(Rattus norvegicus (Rat))
Georgetown University Medical Center

Curated by ChEMBL
LigandPNGBDBM50102113((2R,4R)-4-amino-1-(pyridin-2-ylmethyl)pyrrolidine-...)
Affinity DataEC50:  3.70E+4nMAssay Description:Effective concentration required for agonistic activity at Metabotropic glutamate receptor 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed