TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 64nMAssay Description:Inhibition of recombinant human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in pheophorbide A efflux preincubated for 30 mins foll...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 97nMAssay Description:Inhibition of recombinant human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in pheophorbide A efflux preincubated for 30 mins foll...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 117nMAssay Description:Inhibition of recombinant human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in pheophorbide A efflux preincubated for 30 mins foll...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 123nMAssay Description:Inhibition of recombinant human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in pheophorbide A efflux preincubated for 30 mins foll...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 129nMAssay Description:Inhibition of recombinant human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in pheophorbide A efflux preincubated for 30 mins foll...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 131nMAssay Description:Inhibition of recombinant human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in pheophorbide A efflux preincubated for 30 mins foll...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 208nMAssay Description:Inhibition of recombinant human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in pheophorbide A efflux preincubated for 30 mins foll...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 212nMAssay Description:Inhibition of recombinant human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in pheophorbide A efflux preincubated for 30 mins foll...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 247nMAssay Description:Inhibition of recombinant human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in pheophorbide A efflux preincubated for 30 mins foll...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 251nMAssay Description:Inhibition of recombinant human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in pheophorbide A efflux preincubated for 30 mins foll...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 276nMAssay Description:Inhibition of recombinant human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in pheophorbide A efflux preincubated for 30 mins foll...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of recombinant human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in pheophorbide A efflux preincubated for 30 mins foll...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 311nMAssay Description:Inhibition of recombinant human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in pheophorbide A efflux preincubated for 30 mins foll...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 321nMAssay Description:Inhibition of recombinant human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in pheophorbide A efflux preincubated for 30 mins foll...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 458nMAssay Description:Inhibition of recombinant human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in pheophorbide A efflux preincubated for 30 mins foll...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 511nMAssay Description:Inhibition of recombinant human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in pheophorbide A efflux preincubated for 30 mins foll...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 679nMAssay Description:Inhibition of recombinant human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in pheophorbide A efflux preincubated for 30 mins foll...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 741nMAssay Description:Inhibition of recombinant human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in pheophorbide A efflux preincubated for 30 mins foll...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 3.63E+3nMAssay Description:Inhibition of recombinant human GFP-fused ABCG2 expressed in MDCK2 cells assessed as reduction in pheophorbide A efflux preincubated for 30 mins foll...More data for this Ligand-Target Pair