Compile Data Set for Download or QSAR
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Found 31 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 7601
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM298418(3-(6-amino-1-(4-amino-2-fluorobenzyl)-1H-pyrazolo[...)
Affinity DataKi: <100nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM50176050(8-(3,4-dimethoxystyryl)-1,3-diethyl-7-methyl-1H-pu...)
Affinity DataKi: <100nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM633466(US11806350, Compound 206)
Affinity DataKi: <100nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM633489(3-(6-amino-1-(4-amino-2,6-difluorobenzyl)-1H-pyraz...)
Affinity DataKi: <100nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM633490(3-(6-amino-1-(4-amino-2,6-difluorobenzyl)-1H-pyraz...)
Affinity DataKi: <100nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM633491(3-(6-amino-1-(4-amino-2-fluorobenzyl)-1H-pyrazolo[...)
Affinity DataKi: <100nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM633492(US11806350, Compound 210)
Affinity DataKi: <100nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM633493(3-(6-amino-1-(4-amino-3-(trifluoromethyl)benzyl)-1...)
Affinity DataKi: <100nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM633494(3-(6-amino-1-(2,6-difluorobenzyl)-1H-pyrazolo[3,4-...)
Affinity DataKi: <100nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM298433(US11806350, Compound 204)
Affinity DataKi: <100nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM633515(2-[6-amino-1-[[4-amino-3-(trifluoromethyl)phenyl]m...)
Affinity DataKi: <100nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM633511(6-(6-amino-1-(2,6-difluorobenzyl)-1H-pyrazolo[3,4-...)
Affinity DataKi: <100nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM633507(6-(6-amino-1-(4-amino-3-methylbenzyl)-1H-pyrazolo[...)
Affinity DataKi: <100nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM633503(6-[6-amino-1-[(4-amino-2,6-difluoro-phenyl)methyl]...)
Affinity DataKi: <100nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM633499(6-[6-amino-1-[(4-amino-2-fluoro-phenyl)methyl]pyra...)
Affinity DataKi: <100nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM633495(6-(6-amino-1-(4-aminobenzyl)-1H-pyrazolo[3,4-d]pyr...)
Affinity DataKi:  550nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM633500(2-(6-amino-1-(4-amino-2-fluorobenzyl)-1H-pyrazolo[...)
Affinity DataKi:  550nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM633512(2-(6-amino-1-(2,6-difluorobenzyl)-1H-pyrazolo[3,4-...)
Affinity DataKi:  550nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM633504(2-[6-amino-1-[(4-amino-2,6-difluoro-phenyl)methyl]...)
Affinity DataKi:  550nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM633508(2-(6-amino-1-(4-amino-3-methylbenzyl)-1H-pyrazolo[...)
Affinity DataKi:  550nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM633496(2-(6-amino-1-(4-aminobenzyl)-1H-pyrazolo[3,4-d]pyr...)
Affinity DataKi:  5.50E+3nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM633514(4-[6-amino-1-[(2,6-difluorophenyl)methyl]pyrazolo[...)
Affinity DataKi:  5.50E+3nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM633513(5-(6-amino-1-(2,6-difluorobenzyl)-1H-pyrazolo[3,4-...)
Affinity DataKi:  5.50E+3nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM633509(5-(6-amino-1-(4-amino-3-methylbenzyl)-1H-pyrazolo[...)
Affinity DataKi: >1.00E+4nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM633510(4-(6-amino-1-(4-amino-3-methylbenzyl)-1H-pyrazolo[...)
Affinity DataKi: >1.00E+4nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM633502(4-(6-amino-1-(4-amino-2-fluorobenzyl)-1H-pyrazolo[...)
Affinity DataKi: >1.00E+4nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM633501(5-[6-amino-1-[(4-amino-2-fluoro-phenyl)methyl]pyra...)
Affinity DataKi: >1.00E+4nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM633498(4-(6-amino-1-(4-aminobenzyl)-1H-pyrazolo[3,4-d]pyr...)
Affinity DataKi: >1.00E+4nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM633505(5-[6-amino-1-[(4-amino-2,6-difluoro-phenyl)methyl]...)
Affinity DataKi: >1.00E+4nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM633497(5-(6-amino-1-(4-aminobenzyl)-1H-pyrazolo[3,4-d]pyr...)
Affinity DataKi: >1.00E+4nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ildong Pharmaceutical

US Patent
LigandPNGBDBM633506(4-(6-amino-1-(4-amino-2,6-difluorobenzyl)-1H-pyraz...)
Affinity DataKi: >1.00E+4nMAssay Description:Test compound is weighed, dissolved in DMSO to make a stock solution of 10 mM, diluted with DMSO to prepare working solutions, then 100-fold diluted ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent