Compile Data Set for Download or QSAR
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Found 2 of affinity data with PDB=2E9V
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM15275(7-chloro-3-oxo-8-[(pyridin-4-ylmethyl)amino]-11,17...)
Affinity DataKi:  13nMAssay Description:Inhibition of Chk1More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM15275(7-chloro-3-oxo-8-[(pyridin-4-ylmethyl)amino]-11,17...)
Affinity DataIC50:  13nMAssay Description:Chk1 kinase activity was assayed in reaction buffer containing substrate, enzyme, and inhibitor in the presence of 5uM ATP/[gamma-33P] ATP. 33P incor...More data for this Ligand-Target Pair