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Found 1 of affinity data with PDB=3E37
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Duke University Medical Center

LigandPNGBDBM31424(ethylenediamine scaffold, 5)
Affinity DataIC50:  4.05E+3nMpH: 7.7 T: 2°CAssay Description:In vitro inhibition assay of human PFT was done by measuring the incorporation of [3H] FPP (Amersham Biosciences, Piscataway, NJ) into wild type H-Ra...More data for this Ligand-Target Pair