Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of affinity data with PDB=3HMM
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50293516(2-(6-methylpyridin-2-yl)-N-(pyridin-4-yl)quinazoli...)
Affinity DataIC50:  25nMAssay Description:Inhibition of human ALK5 kinase expressed in Sf9 cellsMore data for this Ligand-Target Pair
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50293516(2-(6-methylpyridin-2-yl)-N-(pyridin-4-yl)quinazoli...)
Affinity DataIC50:  95nMAssay Description:Inhibition of TGFbeta-induced ALK5 in human HepG2 cells by luciferase assayMore data for this Ligand-Target Pair
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50293516(2-(6-methylpyridin-2-yl)-N-(pyridin-4-yl)quinazoli...)
Affinity DataIC50:  6.72E+3nMAssay Description:Inhibition of GST-fused p38alphaMore data for this Ligand-Target Pair