Compile Data Set for Download or QSAR
maximum 50k data
Found 2 of affinity data with PDB=4E4L
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50392018(CHEMBL2152409)
Affinity DataKi:  1.70nMAssay Description:Inhibition of JAK1More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50392018(CHEMBL2152409)
Affinity DataEC50:  210nMAssay Description:Inhibition of JAK1 in human TF1 cells assessed as inhibition of IL2-induced STAT3 phosphorylationMore data for this Ligand-Target Pair