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Found 1 of affinity data with PDB=5ETH
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50161156(CHEMBL3793914)
Affinity DataIC50:  56nMAssay Description:Inverse agonist activity at recombinant human GST-tagged ROR-gamma receptor ligand binding domain assessed as inhibition of receptor and co-activator...More data for this Ligand-Target Pair