Compile Data Set for Download or QSAR
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Found 4 of affinity data with PDB=5JD7
TargetIsoform Beta of cGMP-dependent protein kinase 1 [1-351](Homo sapiens (Human))
Baylor College of Medicine

LigandPNGBDBM65505(PET-cGMP)
Affinity DataEC50:  3.80nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
TargetIsoform Beta of cGMP-dependent protein kinase 1 [5-676,G306E](Homo sapiens (Human))
Baylor College of Medicine

LigandPNGBDBM65505(PET-cGMP)
Affinity DataEC50:  18nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
TargetIsoform Beta of cGMP-dependent protein kinase 1 [1-351,G306E](Homo sapiens (Human))
Baylor College of Medicine

LigandPNGBDBM65505(PET-cGMP)
Affinity DataEC50: <2nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair
TargetIsoform Beta of cGMP-dependent protein kinase 1 [1-351,G182E](Homo sapiens (Human))
Baylor College of Medicine

LigandPNGBDBM65505(PET-cGMP)
Affinity DataEC50:  5.80nMpH: 7.0Assay Description:Kinase activity was determined employing a microfluidic mobility-shift assay on a Caliper DeskTop Profiler (Caliper Life Sciences, PerkinElmer). The ...More data for this Ligand-Target Pair