Compile Data Set for Download or QSAR
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Found 2 of affinity data with PDB=5LWP
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Galderma R & D

Curated by ChEMBL
LigandPNGBDBM50203462(CHEMBL3931161)
Affinity DataIC50:  31nMAssay Description:Inverse agonist activity at GAL4 DBD-fused RORgammat LBD (unknown origin) expressed in HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Galderma R & D

Curated by ChEMBL
LigandPNGBDBM50203462(CHEMBL3931161)
Affinity DataIC50:  40nMAssay Description:Inverse agonist activity at RORgamma in human CD4+ T cells assessed as inhibition of IL-17A release after 4 days by HTRF assayMore data for this Ligand-Target Pair