Affinity DataIC50: 3.16E+5nMAssay Description:Binding constant against dopamine receptor D2 (in vitro)More data for this Ligand-Target Pair
Affinity DataIC50: 3.19E+5nMAssay Description:Inhibition of recombinant human N-terminal His-tagged KHK expressed in Escherichia coli BL21(DE3) using fructose as substrate incubated for 30 mins f...More data for this Ligand-Target Pair
Affinity DataKd: 6.20E+4nMAssay Description:Binding affinity to full length recombinant human biotin-labeled KHK by SPR assayMore data for this Ligand-Target Pair