TargetMu-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania
Curated by PDSP Ki Database
University of Pennsylvania
Curated by PDSP Ki Database
TargetMu-type opioid receptor(MOUSE)
Memorial Sloan-Kettering Cancer Center
Curated by PDSP Ki Database
Memorial Sloan-Kettering Cancer Center
Curated by PDSP Ki Database
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania
Curated by PDSP Ki Database
University of Pennsylvania
Curated by PDSP Ki Database
TargetMu-type opioid receptor(MOUSE)
Memorial Sloan-Kettering Cancer Center
Curated by PDSP Ki Database
Memorial Sloan-Kettering Cancer Center
Curated by PDSP Ki Database
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania
Curated by PDSP Ki Database
University of Pennsylvania
Curated by PDSP Ki Database
Affinity DataKi: 1.10nMAssay Description:Binding affinity to mu opioid receptor (unknown origin) expressed in HEK cells at pH 7.4More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Pennsylvania
Curated by PDSP Ki Database
University of Pennsylvania
Curated by PDSP Ki Database
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Pennsylvania
Curated by PDSP Ki Database
University of Pennsylvania
Curated by PDSP Ki Database
Affinity DataKi: 1.5nMAssay Description:Binding affinity of compound evaluated for Opioid receptor mu 1 isolated from rat brainMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania
Curated by PDSP Ki Database
University of Pennsylvania
Curated by PDSP Ki Database
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Pennsylvania
Curated by PDSP Ki Database
University of Pennsylvania
Curated by PDSP Ki Database
Affinity DataKi: 2.20nMAssay Description:Displacement [3H]-naloxone from the Opioid receptor mu 1 isolated from rat brain membrane.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Pennsylvania
Curated by PDSP Ki Database
University of Pennsylvania
Curated by PDSP Ki Database
Affinity DataKi: 2.20nMAssay Description:Ability to displace [3H]-naloxone from the Opioid receptor mu 1 isolated from the rat brain membranes.More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania
Curated by PDSP Ki Database
University of Pennsylvania
Curated by PDSP Ki Database
Affinity DataKi: 2.90nMAssay Description:Displacement of [3H]-DAMGO (2 nM ) from opioid receptor mu 1 in human brainMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Pennsylvania
Curated by PDSP Ki Database
University of Pennsylvania
Curated by PDSP Ki Database
Affinity DataKi: 4nMAssay Description:Binding affinity towards Opioid receptor mu 1 using [3H]DAMGO as radioligand.More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania
Curated by PDSP Ki Database
University of Pennsylvania
Curated by PDSP Ki Database
Affinity DataKi: 4nMAssay Description:Binding affinity against Opioid receptor mu 1More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Pennsylvania
Curated by PDSP Ki Database
University of Pennsylvania
Curated by PDSP Ki Database
Affinity DataKi: 5.90nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(MOUSE)
Memorial Sloan-Kettering Cancer Center
Curated by PDSP Ki Database
Memorial Sloan-Kettering Cancer Center
Curated by PDSP Ki Database
Affinity DataKi: 5.90nMAssay Description:Displacement of [3H]-DAMGO from Swiss Webster mouse neural membranes mu opioid receptor after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Pennsylvania
Curated by PDSP Ki Database
University of Pennsylvania
Curated by PDSP Ki Database
Affinity DataKi: 5.90nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Pennsylvania
Curated by PDSP Ki Database
University of Pennsylvania
Curated by PDSP Ki Database
Affinity DataKi: 570nMAssay Description:Displacement of [3H] DAMGO from rat mu-opioid receptorMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Binding affinity to opioid receptors by the displacement of [3H]fentanyl in rat brain homogenatesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania
Curated by PDSP Ki Database
University of Pennsylvania
Curated by PDSP Ki Database
Affinity DataIC50: 1.30nMAssay Description:Binding affinity against mu-opiate receptor (human) using [3H]DAMGO radioligandMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Displacement [3H]naloxone from rat-brain Opioid receptorsMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania
Curated by PDSP Ki Database
University of Pennsylvania
Curated by PDSP Ki Database
Affinity DataIC50: 5.5nMAssay Description:Agonist activity at Gi-coupled mu opioid receptor (unknown origin) expressed in HEK293T cells assessed as inhibition of cAMP production at pH 6.5 mea...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania
Curated by PDSP Ki Database
University of Pennsylvania
Curated by PDSP Ki Database
Affinity DataIC50: 11nMAssay Description:Agonist activity at Gi-coupled mu opioid receptor (unknown origin) expressed in HEK293T cells assessed as inhibition of cAMP production at pH 7.4 mea...More data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Displacement of [3H]nalotrexone from rat-brain Opioid receptorsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:In vivo binding affinity to opioid receptor preparations from rat brainMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Pennsylvania
Curated by PDSP Ki Database
University of Pennsylvania
Curated by PDSP Ki Database
Affinity DataIC50: 1.26E+3nMAssay Description:Displacement of [3H] DAMGO from rat mu-opioid receptorMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania
Curated by PDSP Ki Database
University of Pennsylvania
Curated by PDSP Ki Database
Affinity DataEC50: 17nMAssay Description:Agonist activity at mu opioid receptor (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation ...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania
Curated by PDSP Ki Database
University of Pennsylvania
Curated by PDSP Ki Database
Affinity DataEC50: 17nMAssay Description:Agonist activity at mu opioid receptor (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation ...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania
Curated by PDSP Ki Database
University of Pennsylvania
Curated by PDSP Ki Database
Affinity DataEC50: 43nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO cell membranes after 1 hr by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania
Curated by PDSP Ki Database
University of Pennsylvania
Curated by PDSP Ki Database
Affinity DataEC50: 53nMAssay Description:Agonist activity at human mu opioid receptor expressed in human U2OS cells co-transfected with beta-arrestin-2 assessed as increase in beta-arrestin-...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Pennsylvania
Curated by PDSP Ki Database
University of Pennsylvania
Curated by PDSP Ki Database
Affinity DataEC50: 0.510nMAssay Description:Agonist activity at human MOR expressed in CHO-K1 cells assessed as cAMP accumulation incubated for 30 mins and measured after 1 hr by Eu-cAMP tracer...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Pennsylvania
Curated by PDSP Ki Database
University of Pennsylvania
Curated by PDSP Ki Database
Affinity DataEC50: 32nMAssay Description:Compound was tested for its ability to stimulate [35S]GTP-gamma-S, binding to membranes from C6 glioma cells stably expressing rat mu opioid receptorMore data for this Ligand-Target Pair