Compile Data Set for Download or QSAR
maximum 50k data
Found 12 of affinity data with PDB=8T1F
TargetTransient receptor potential cation channel subfamily V member 4(Mus musculus)
Kunming University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50192821(CHEMBL2133556)
Affinity DataIC50:  17nMAssay Description:Antagonist activity at mouse TRPV4More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Mus musculus)
Kunming University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50192821(CHEMBL2133556)
Affinity DataIC50:  17nMAssay Description:Antagonist activity at mouse TRPV4 expressed in HEK293 cells assessed as inhibition of 4alpha-PDD-induced current at holding potential of -40 mV by W...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Kunming University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50192821(CHEMBL2133556)
Affinity DataIC50:  18nMAssay Description:Antagonist activity at human TRPV4More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Kunming University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50192821(CHEMBL2133556)
Affinity DataIC50:  29nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of hypotonicity-induced activation pretreated for 5 mi...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Kunming University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50192821(CHEMBL2133556)
Affinity DataIC50:  48nMAssay Description:Antagonist activity at TRPV4 (unknown origin)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Kunming University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50192821(CHEMBL2133556)
Affinity DataIC50:  48nMAssay Description:Antagonist activity at human TRPV4 expressed in HEK293 cells assessed as inhibition of 4alpha-PDD-induced current at holding potential of -40 mV by W...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Kunming University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50192821(CHEMBL2133556)
Affinity DataIC50:  57nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Kunming University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50192821(CHEMBL2133556)
Affinity DataIC50:  57nMAssay Description:Antagonist activity at human TRPV4 assessed as inhibition of 4alpha-PDD-induced activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Kunming University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50192821(CHEMBL2133556)
Affinity DataIC50:  57nMAssay Description:Antagonist activity at human recombinant TRPV4 expressed in CHO-K1 cells assessed as blockade of 1000 nM 4alphaPDD-induced calcium mobilization by FL...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Rattus norvegicus)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50192821(CHEMBL2133556)
Affinity DataIC50:  133nMAssay Description:Antagonist activity at rat TRPV4 expressed in HEK293 cells assessed as inhibition of 4alpha-PDD-induced current at holding potential of -40 mV by Who...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Rattus norvegicus)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50192821(CHEMBL2133556)
Affinity DataIC50:  133nMAssay Description:Antagonist activity at rat TRPV4More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Rattus norvegicus)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50192821(CHEMBL2133556)
Affinity DataIC50:  180nMAssay Description:Antagonist activity at recombinant rat TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins fo...More data for this Ligand-Target Pair