Affinity DataIC50: 2.40nMAssay Description:Binding affinity towards Nicotinic acetylcholine receptor by the displacement of [3H]-nicotine from rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Binding affinity towards Nicotinic acetylcholine receptor by the displacement of [3H]-nicotine from rat cortical membranesMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-9(Homo sapiens (Human))
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
The Danish University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibitory concentration against Nicotinic acetylcholine receptor alpha9; Range is 100-200 nMMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+4nMAssay Description:The compound was tested for inhibitory potency against Nicotinic acetylcholine receptor in Rat muscle.More data for this Ligand-Target Pair