Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) for PDB: 10AD
TargetCalcium-activated potassium channel subunit alpha-1(Rat)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347497BDBM50347497(CHEMBL384903)
Affinity DataIC50: 4.37E+3nMAssay Description:Induction of BK channel mediated vasorelaxation activity in Kcl-induced contraction in Wistar rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCalcium-activated potassium channel subunit alpha-1(Rat)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347497BDBM50347497(CHEMBL384903)
Affinity DataIC50: 5.01E+3nMAssay Description:Activation of large-conductance calcium-activated potassium channel-mediated vasorelaxation in endothelium-denuded normotensive Wistar rat thoracic a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCalcium-activated potassium channel subunit alpha-1(Rat)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347497BDBM50347497(CHEMBL384903)
Affinity DataIC50: 5.13E+3nMAssay Description:Activation of BK channel in Wistar rat thoracic aorta assessed as relaxation of KCl-induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCalcium-activated potassium channel subunit alpha-1(Human)
University of Pisa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347497BDBM50347497(CHEMBL384903)
Affinity DataIC50: 5.89E+3nMAssay Description:Activation of BK channel-mediated vasorelaxation activity assessed as reduction in KCl-induced contractile toneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)