Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 3VSP
TargetPeroxisome proliferator-activated receptor gamma(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50050557(CHEMBL3317858)
Affinity DataKd:  2.90nMAssay Description:Binding affinity to human His-tagged PPARgamma LBD by SPR methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor gamma(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50050557(CHEMBL3317858)
Affinity DataEC50:  53nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)