Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) for PDB: 3WQH
TargetDipeptidyl peptidase 4(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50359366(CHEMBL1929387 | CHEMBL1929396 | US20240115577, Com...)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of human DPP4 expressed in Silkworm baculovirus system preincubated for 30 mins followed by substrate addition and measured after 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetDipeptidyl peptidase 4(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50359366(CHEMBL1929387 | CHEMBL1929396 | US20240115577, Com...)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of human recombinant DPP-4 using H-Gly-Pro-AMC as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetDipeptidyl peptidase 4(Human)
Tianjin University

Curated by ChEMBL
LigandPNGBDBM50359366(CHEMBL1929387 | CHEMBL1929396 | US20240115577, Com...)
Affinity DataIC50: 11.4nMAssay Description:Human DPP4 activity assay data were obtained using a DPP4 Activity Assay Kit (Sigma-Aldrich, MAK088) according to the manufacturer's instructions...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2024
Entry Details
US Patent
PDB3D3D Structure (crystal)