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Found
1
Enz. Inhib. hit(s) for PDB:
4AN9
Target
Dual specificity mitogen-activated protein kinase kinase 1
(Human)
TBA
Curated by
ChEMBL
Ligand
BDBM50391809
(CHEMBL2146887)
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Affinity Data
IC50: 44nM
Assay Description:
Inhibition of MEK1-mediated ERK2 T202/Y204 phosphorylation using biotinylated MBP as substrate preincubated for 30 mins measured after 100 mins by cR...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
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Ligand Info
CHEMBL
PC cid
PC sid
PDB
Similars
In Depth
Date in BDB:
5/17/2013
Entry Details
Article
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PubMed
PDB
3D Structure (crystal)
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