Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) for PDB: 4C7T
TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438033(CHEMBL2409605)
Affinity DataIC50: 400nMAssay Description:Inhibition of pre-activated recombinant full length FAK (unknown origin) using ULight labeled poly(Glu/Tyr) as substrate after 1.6 hrs by TR-FRET ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438033(CHEMBL2409605)
Affinity DataIC50: 400nMAssay Description:Inhibition of FAK (unknown origin) using ULight-poly GT as substrate after 1.6 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/2/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetFocal adhesion kinase 1(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50438033(CHEMBL2409605)
Affinity DataIC50: 400nMAssay Description:Inhibition of FAK (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMedPDB3D3D Structure (crystal)