Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 4JVI
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Pharmaceutical and Drug Industries Research Institute

Curated by ChEMBL
LigandPNGBDBM50512170(CHEMBL4518045)
Affinity DataIC50: 1.20E+3nMAssay Description:Antagonist activity at PqsR in wild-type Pseudomonas aeruginosa PAO1-LMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetVirulence factor transcriptional regulator MvfR(Pseudomonas aeruginosa)
Pharmaceutical and Drug Industries Research Institute

Curated by ChEMBL
LigandPNGBDBM50512170(CHEMBL4518045)
Affinity DataIC50: 5.00E+3nMAssay Description:Antagonist activity at His6 -tagged Pseudomonas aeruginosa PqsR CBD domain expressed in Escherichia coli Rosetta 2 (DE3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)