Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) for PDB: 4NRA
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495371(CHEMBL3110247)
Affinity DataIC50: 2.40E+4nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495371(CHEMBL3110247)
Affinity DataIC50: 3.70E+4nMAssay Description:Displacement of biotinylated H3Kac14 peptide from His6-tagged human BAZ2B expressed in Escherichia coli BL21(DE3) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
University of Cambridge

Curated by ChEMBL
LigandPNGBDBM50495371(CHEMBL3110247)
Affinity DataKd:  6.50E+4nMAssay Description:Binding affinity to human BAZ2B expressed in Escherichia coli BL21(DE3) by competitive isothermal titration calorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)