Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 4RMD
TargetRetinoic acid receptor RXR-alpha(Human)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50123614(CHEMBL3622723)
Affinity DataEC50:  19nMAssay Description:Agonist activity at human RXRalpha LBD expressed in HEK293 cells transfected with Gal4 reporter assessed as increase of transcription by dual lucifer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetRetinoic acid receptor RXR-alpha(Human)
University of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50123614(CHEMBL3622723)
Affinity DataKd:  35nMAssay Description:Binding affinity to human RXRalpha LBD by fluorescence quenching methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)