Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) for PDB: 4TS8
TargetCREB-binding protein(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50172107(CHEMBL3810303)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of CREBBP (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCREB-binding protein(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50172107(CHEMBL3810303)
Affinity DataKd:  2.00E+4nMAssay Description:Competitive binding affinity to human His-tagged CREBBP (1081 to 1097 residues) expressed in T7 phage-infected Escherichia coli BL21(DE3) cells measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCREB-binding protein(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50172107(CHEMBL3810303)
Affinity DataKd:  2.00E+4nMAssay Description:Competitive binding affinity to CBP (unknown origin) measured after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)