Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) for PDB: 5APH
TargetNuclear receptor ROR-gamma(Human)
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50534854(CHEMBL4544537)
Affinity DataIC50: 60nMAssay Description:Agonist activity at human RORgammatMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetNuclear receptor ROR-gamma(Human)
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50534854(CHEMBL4544537)
Affinity DataIC50: 60nMAssay Description:Displacement of [3H]T0901317 from N-6HN-MBP-Avi-TCS-tagged human RORgamma LBD (P260 to K518 residues) preincubated for 30 mins followed by ligand add...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNuclear receptor ROR-gamma(Human)
Southern Medical University

Curated by ChEMBL
LigandPNGBDBM50534854(CHEMBL4544537)
Affinity DataIC50: 60nMAssay Description:Agonist activity at ROR gamma (unknown origin) by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMedPDB3D3D Structure (crystal)