Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) for PDB: 5B0X
TargetCasein kinase II subunit alpha'(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50420563(CHEMBL2087023)
Affinity DataIC50: 11nMAssay Description:Inhibition of GST-tagged human CK2alpha' (1 to 350 residues) using CK2tide as substrate incubated for 1 hr by off-chip mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50420563(CHEMBL2087023)
Affinity DataIC50: 20nMAssay Description:Inhibition of GST-tagged human CK2alpha (1 to 391 residues) using CK2tide as substrate incubated for 1 hr by off-chip mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50420563(CHEMBL2087023)
Affinity DataIC50: 20nMAssay Description:Inhibition of human CK2alpha (2 to 391 residues) using [33P]-ATP by scintillation counting based radioactive filter binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50420563(CHEMBL2087023)
Affinity DataIC50: 32nMAssay Description:Competitive inhibition of GST fused human CK2alpha expressed in Escherichia coli BL21 after 10 mins in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha'(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50420563(CHEMBL2087023)
Affinity DataIC50: 46nMAssay Description:Competitive inhibition of GST fused human CK2alpha' expressed in Escherichia coli BL21 after 10 mins in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)