Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 5HJS
TargetOxysterols receptor LXR-alpha(Human)
Wuxi Apptec

Curated by ChEMBL
LigandPNGBDBM50172521(CHEMBL3809850)
Affinity DataEC50:  420nMAssay Description:Partial agonist activity at GST-tagged LXRalpha-LBD (unknown origin) by LanthaScreen TR-FRET liver X receptor coactivator assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetOxysterols receptor LXR-alpha(Human)
Wuxi Apptec

Curated by ChEMBL
LigandPNGBDBM50172521(CHEMBL3809850)
Affinity DataEC50:  830nMAssay Description:Partial agonist activity at LXRalpha (unknown origin) expressed in human HepG2 cells co-expressing ABCA1 promoter measured after 48 hrs by cell-based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)