Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 5JGD
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Chugai Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187111(CHEMBL3823738)
Affinity DataIC50: 11nMAssay Description:Inhibition of GST-tagged TAK1 (unknown origin) expressed in sf9 cells coexpressing His-tagged TAB1 using myelin basic protein as substrate incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50187111(CHEMBL3823738)
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant human full-length His-tagged TAK1-TAB1 fusion protein (437 to 504 residues) expressed in baculovirus expression system usin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)