Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 5K0X
TargetTyrosine-protein kinase Mer(Human)
Unc Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM308455(US9649309, Compound UNC2541A)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of MERTK (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTyrosine-protein kinase Mer(Human)
Unc Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM308455(US9649309, Compound UNC2541A)
Affinity DataIC50: 10nMAssay Description:Briefly, activity assays were performed in a 384 well, polypropylene microplate in a final volume of 50 μL of 50 mM Hepes, Ph 7.4 containing 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
US Patent
PDB3D3D Structure (crystal)