Compile Data Set for Download or QSAR
Report error Found 1 Enz. Inhib. hit(s) for PDB: 5KKR
TargetKinase suppressor of Ras 2(Human)
Icahn School of Medicine At Mount Sinai

US Patent
LigandPNGBDBM429286(APS-2-79 | US10548897, Compound 21)
Affinity DataIC50: 120nMAssay Description:The ATP-biotin assay was performed in buffer containing 25 mM Tris pH 7.5, 150 mM NaCl, 10 mM MgCl2, and 2% DMSO. Purified hKSR2-rMEK1 was assayed at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent
PDB3D3D Structure (crystal)