Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 5L0E
TargetAutotaxin(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50535214BDBM50535214(CHEMBL4549771)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of recombinant full length human C-terminal His-tagged autotaxin expressed in human 293E cells assessed as choline release using lysophosp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAutotaxin(Human)
Lilly Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50535214BDBM50535214(CHEMBL4549771)
Affinity DataIC50: 42nMAssay Description:Inhibition of autotaxin in healthy human plasma assessed as reduction in LPA level after 3 hrs by mass spectrometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)