Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 5MJ6
TargetLeucyl-cystinyl aminopeptidase(Human)
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50236826(CHEMBL4065841)
Affinity DataKi:  18nMAssay Description:Inhibition of recombinant human IRAP expressed in GnT1 deficient HEK293S cells using L-leucine 7-amido-4-methyl coumarin as substrate after 5 to 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetLeucyl-cystinyl aminopeptidase(Human)
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50236826(CHEMBL4065841)
Affinity DataIC50: 32nMAssay Description:Inhibition of IRAP (unknown origin) expressed in HEK 293S GnTI(-) cells by in vitro fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)