Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) for PDB: 5W5V
TargetSerine/threonine-protein kinase TBK1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM357857(US10214536, Amlexanox | Aphthasol)
Affinity DataIC50: 850nMAssay Description:Inhibition of human TBK1 (1 to 657 residues) expressed in Baculovirus infected SF9 insect cells using myelin basic protein as substrate in presence o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase TBK1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM357857(US10214536, Amlexanox | Aphthasol)
Affinity DataIC50: 851nMAssay Description:Inhibition of human TBK1 (1 to 657 residues) expressed in Baculovirus infected SF9 insect cells using myelin basic protein as substrate in presence o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase TBK1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM357857(US10214536, Amlexanox | Aphthasol)
Affinity DataIC50: 980nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent
PDB3D3D Structure (crystal)