Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) for PDB: 6B4U
LigandPNGBDBM50078154(CHEMBL3417694)
Affinity DataKi:  9nMAssay Description:Displacement of fluorescent labeled NOXA peptide from recombinant human MCL1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50078154(CHEMBL3417694)
Affinity DataKi:  21nMAssay Description:Displacement of F-Bak (GQVGRQLAIIGDK(6-FAM)INR-amide) from MCL1 (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50078154(CHEMBL3417694)
Affinity DataKi:  190nMAssay Description:Binding affinity to Mcl-1 (unknown origin) pre-incubated for 30 mins followed by addition FAM-peptide further incubated for 20 mins by fluorescence p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50078154(CHEMBL3417694)
Affinity DataKi:  470nMAssay Description:Displacement of fluorescent labeled NOXA peptide from recombinant human MCL1 by fluorescence polarization assay in presence of 1% human serumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50078154(CHEMBL3417694)
Affinity DataKi:  1.23E+3nMAssay Description:Displacement of F-Bak (GQVGRQLAIIGDK(6-FAM)INR-amide) from MCL1 (unknown origin) after 1 hr by TR-FRET assay in presence of 10% human serumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)