Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) for PDB: 6P69
TargetFibroblast growth factor receptor 1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM249404(US9434697, 121 | US9730931, Compound 121 | US10537...)
Affinity DataIC50: 1.02E+3nMAssay Description:Recombinant FGFR1 (2.5 nM), FGFR2 (1 nM), FGFR3 (5 nM), or FGFR4 (12 nM) (Invitrogen™) was prepared as a mixture with substrate KKKSPGEYVNIEFG (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2019
Entry Details
US Patent
PDB3D3D Structure (crystal)
TargetFibroblast growth factor receptor 1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM249404(US9434697, 121 | US9730931, Compound 121 | US10537...)
Affinity DataIC50: 1.02E+3nMAssay Description:Recombinant FGFR1 (2.5 nM), FGFR2 (1 nM), FGFR3 (5 nM), or FGFR4 (12 nM) was prepared as a mixture with substrate KKKSPGEYVNIEFG (SEQ ID NO:1) (20 M,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2020
Entry Details
US Patent
PDB3D3D Structure (crystal)
TargetFibroblast growth factor receptor 1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM249404(US9434697, 121 | US9730931, Compound 121 | US10537...)
Affinity DataIC50: 1.02E+3nMAssay Description:Recombinant FGFR1 (2.5 nM), FGFR2 (1 nM), FGFR3 (5 nM), or FGFR4 (12 nM) (Invitrogen ) was prepared as a mixture with substrate KKKSPGEYVNIEFG (SEQ I...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2021
Entry Details
US Patent
PDB3D3D Structure (crystal)
TargetFibroblast growth factor receptor 1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM249404(US9434697, 121 | US9730931, Compound 121 | US10537...)
Affinity DataIC50: 1.02E+3nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
US Patent
PDB3D3D Structure (crystal)