Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 6VIF
TargetNuclear receptor subfamily 5 group A member 2(Human)
Emory University

Curated by ChEMBL
LigandPNGBDBM50544057(CHEMBL4637563)
Affinity DataKi:  38nMAssay Description:Displacement of 6N-FAM from human LRH1 LBD (299 to 541 residues) expressed in Escherichia coli BL21 pLysS by competitive binding based fluorescence p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNuclear receptor subfamily 5 group A member 2(Human)
Emory University

Curated by ChEMBL
LigandPNGBDBM50544057(CHEMBL4637563)
Affinity DataEC50:  400nMAssay Description:Agonist activity at LRH1 (unknown origin) by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)