Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 6ZLY
TargetPeroxisome proliferator-activated receptor gamma(Human)
Aix Marseille University

Curated by ChEMBL
LigandPNGBDBM50554670(CHEMBL4741141)
Affinity DataKd:  94nMAssay Description:Binding affinity to PPARg (unknown origin) by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor gamma(Human)
Aix Marseille University

Curated by ChEMBL
LigandPNGBDBM50554670(CHEMBL4741141)
Affinity DataEC50:  1.94E+3nMAssay Description:Agonist activity at GAL4-tagged PPARg-LBD (unknown origin) expressed in HEK293 cells assessed as induction of receptor transactivation incubated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)