Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 7E2E
TargetSteroid hormone receptor ERR1(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50557798(CHEMBL4760865)
Affinity DataIC50: 800nMAssay Description:Inhibition of FITC-RIP140 peptide binding to N-terminal His-tagged human GST-ERRalpha-LBD (290 to 519 residues) expressed in Escherichia coli incubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSteroid hormone receptor ERR1(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50557798(CHEMBL4760865)
Affinity DataEC50:  5.40E+3nMAssay Description:Agonist activity at recombinant full-length human ERRalpha expressed in MG63 cells assessed as transcriptional activation incubated for 18 hrs by dua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)