Affinity DataKi: 2.20nMAssay Description:Binding affinity to human 5-HT1F assessed as inhibition constant incubated for 10 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 88nMAssay Description:Agonist activity at 5HT1F receptor (unknown origin) expressed in HEK293 cells measured after 60 mins by Fluo-4AM dye based FLIPR assayMore data for this Ligand-Target Pair

3D Structure (crystal)