TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of recombinant DYRK1A (unknown origin) using DYRKtide as substrate incubated for 2 hrs in presence of ATP by ADP-Glo kinase assayMore data for this Ligand-Target Pair

3D Structure (crystal)