Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) for PDB: 7M3G
TargetExtracellular calcium-sensing receptor(Rat)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50272591(CHEMBL4128835)
Affinity DataIC50: 31nMAssay Description:Agonist activity at CaSR in rat parathyroid cells assessed as inhibition of PTH (1 to 84 residues) production in presence of Cacl2 by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetExtracellular calcium-sensing receptor(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50272591(CHEMBL4128835)
Affinity DataEC50:  93nMAssay Description:Agonist activity at human CaSR expressed in CHO cells assessed as increase in intracellular calcium mobilization after 1 hr by Fura-2 dye-based fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)