Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) for PDB: 7Q52
TargetSerine/threonine-protein kinase PknG(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidad De Buenos Aires

Curated by ChEMBL
LigandPNGBDBM50600797(CHEMBL5183885)
Affinity DataKd:  2.00E+3nMAssay Description:Binding affinity to full length Mycobacterium tuberculosis protein kinase G expressed in Escherichia coli BL21 assessed as dissociation constant at 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase PknG(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidad De Buenos Aires

Curated by ChEMBL
LigandPNGBDBM50600797(CHEMBL5183885)
Affinity DataKd:  2.20E+3nMAssay Description:Binding affinity to full length Mycobacterium tuberculosis protein kinase G expressed in Escherichia coli BL21 assessed as dissociation constant at 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase PknG(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidad De Buenos Aires

Curated by ChEMBL
LigandPNGBDBM50600797(CHEMBL5183885)
Affinity DataKd:  3.60E+3nMAssay Description:Binding affinity to full length Mycobacterium tuberculosis protein kinase G expressed in Escherichia coli BL21 assessed as apparent dissociation cons...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase PknG(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universidad De Buenos Aires

Curated by ChEMBL
LigandPNGBDBM50600797(CHEMBL5183885)
Affinity DataKd:  8.10E+3nMAssay Description:Binding affinity to full length Mycobacterium tuberculosis protein kinase G expressed in Escherichia coli BL21 assessed as change in melting temperat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMedPDB3D3D Structure (crystal)