Affinity DataKi: 38nMAssay Description:Inhibition of HHAT (unknown origin) assessed as inhibition constant by Pal-CoA Competitive assayMore data for this Ligand-Target Pair
Affinity DataIC50: 76nMAssay Description:Inhibition of HHAT in human HEK293a SHH+ cells assessed as inhibition SHH-YnPal tagging measured after 7 hrs by cell-based tagging assayMore data for this Ligand-Target Pair
Affinity DataIC50: 76nMAssay Description:Inhibition of HHAT in human HEK293a SHH+ cells assessed as inhibition SHH-YnPal tagging measured after 7 hrs by cell-based tagging assayMore data for this Ligand-Target Pair
Affinity DataEC50: 99nMAssay Description:Inhibition of HHAT in human HEK293a SHH+ cells incubated with compound for 24 hrs followed by transferred into SHH-Light2 cells cellular incubated fo...More data for this Ligand-Target Pair
Affinity DataIC50: 750nMAssay Description:Inhibition of human recombinant HHAT using SHH-FAM peptide as substrate for 30 mins by acylation coupled lipophilic induction of polarization (acyl-c...More data for this Ligand-Target Pair
Affinity DataIC50: 750nMAssay Description:Inhibition of HHAT (unknown origin)More data for this Ligand-Target Pair

3D Structure (crystal)