Affinity DataIC50: 3.16nMAssay Description:Inhibition of AChE by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataKi: 6.90nM ΔG°: -46.1kJ/molepH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Estimates of the competitive inhibition constants (Ki) were ob...More data for this Ligand-Target Pair
Affinity DataIC50: 7.5nMAssay Description:Inhibition of AChE (unknown origin) using acetylcholine iodate as substrate preincubated for 10 mins followed by substrate addition by Ellman's metho...More data for this Ligand-Target Pair
Affinity DataKi: 7.64nM IC50: 7.53nMpH: 8.0Assay Description:AChI and 5,5'-dithio-bis(2-nitro-benzoic)acid (DTNB) were used as substrate for this enzymatic reaction. To this end, 100 µL of Tris/HCl buffer (...More data for this Ligand-Target Pair
Affinity DataKi: 7.60nMAssay Description:Inhibition of AChE (unknown origin) using acetylcholine iodate as substrate preincubated for 10 mins followed by substrate addition by Lineweaver-Bur...More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant human AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured...More data for this Ligand-Target Pair
Affinity DataKd: 18nMAssay Description:Dissociation constant towards Acetylcholinesterase in mouseMore data for this Ligand-Target Pair
Affinity DataKi: 18nM ΔG°: -44.2kJ/molepH: 7.0 T: 2°CAssay Description:Assays were conducted at 25 C in 20 mM sodium phosphate buffer (pH 7.0) and 0.01% bovine serum albumin unless otherwise noted. AChE concentrations we...More data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Inhibition of human erythrocyte AChE using ATC iodide as substrate preincubated for 4.5 mins followed by substrate addition measured after 2.5 mins b...More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of human erythrocyte AChE using ATC iodide as substrate preincubated for 4.5 mins followed by substrate addition measured after 2.5 mins b...More data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Inhibition of AChE (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Displacement of propidium iodide from AChE in bovine erythrocytes after 15 mins by fluorescence plate readerMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of human acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibitory activity against acetylcholinesterase in human RBCMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate incubated for 5 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibition of AChE in Swiss Webster mouse cerebral homogenate using acetylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:In vitro inhibitory activity against human erythrocyte acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibition of mouse brain AChEMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibition of acetylcholinesterase (AChE) of human red blood cell (type XIII) by modified radiometric AChE assayMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Inhibition of human recombinant AChEMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Inhibition of human recombinant AChEMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysisMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Inhibition of fetal Bovine serum AChEMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of AChE in bovine erythrocyte by Ellman methodMore data for this Ligand-Target Pair
Affinity DataKi: 40nM ΔG°: -42.2kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition of enzyme activity was measured over a substrate concentration range of 0.01-30 mM and at least six inhibitor concentrations to determine ...More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of bovine erythrocyte AChE by Ellman's reactionMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of bovine erythrocytes AChE by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The absorbance changes at 412 nm were recorded for 5 min with ...More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of bovine erythrocyte AChE by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataKi: 40nM ΔG°: -42.2kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition of enzyme activity was measured over a substrate concentration range of 0.01-30 mM and at least six inhibitor concentrations to determine ...More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of AChE in bovine erythrocytes using acetylthiocholine as substrate by Ellman methodMore data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:Inhibition of AChE (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 45.1nMAssay Description:Inhibition of AChE by Ellman's assayMore data for this Ligand-Target Pair
Affinity DataIC50: 46nMAssay Description:Inhibition of Acetylcholinesterase in rat red blood cellMore data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:Inhibition of human plasma BChEMore data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:Inhibition of human erythrocytes BChEMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:In vitro inhibitory activity against acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 55nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 56nMpH: 8.0 T: 2°CAssay Description:Suitable agents like donepezil hydrochloride and tacrine hydrochloride hydrate were used as standards for this study. Buffer solution (50 mM Tris-HCl...More data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:In vitro inhibitory effect on rat AcetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 72nMAssay Description:Inhibition of human erythrocytes AChE by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 72nMAssay Description:Inhibition of human AChEMore data for this Ligand-Target Pair
Affinity DataIC50: 72nMAssay Description:Inhibition of human AChEMore data for this Ligand-Target Pair
Affinity DataIC50: 75nMAssay Description:Inhibition of Acetylcholinesterase in monkey red blood cellMore data for this Ligand-Target Pair
Affinity DataIC50: 76nMAssay Description:Inhibitory activity against AcetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 76.0nMAssay Description:Inhibition acetylcholinesterase (AChE) enzyme.More data for this Ligand-Target Pair
Affinity DataIC50: 77nMAssay Description:Inhibition of human AChE pre-incubated for 6 mins before ATCI substrate addition and measured after 12 mins by DTNB reagent dependent UV-Vis spectrop...More data for this Ligand-Target Pair
Affinity DataIC50: 77nMAssay Description:Inhibition of human AChE by Ellman's assayMore data for this Ligand-Target Pair

3D Structure (crystal)