Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) for PDB: 8BGC
TargetCasein kinase II subunit alpha'(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50614163(CHEMBL5288779)
Affinity DataIC50: 200nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha' expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K5 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50614163(CHEMBL5288779)
Affinity DataIC50: 920nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K10 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha'(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50614163(CHEMBL5288779)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of wild type human CK2alpha' in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50614163(CHEMBL5288779)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of wild type human CK2alpha in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMedPDB3D3D Structure (crystal)